IMG-EN-AS-60869-01.jpg
Peptides

Cetrorelix Acetate, Cetrotide - 1 mg

$195.00
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  • Cat.Number : AS-60869
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    In stock

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A highly modified luteinizing hormone-releasing hormone (LHRH) decapeptide with a terminal amide group, this peptide is a LHRH antagonist. It regulates the expression of Galphas and Galphai protein subunits and adenylate cyclase activity in ovary, breast and pituitary. Cetrorelix competitively inhibits LHRH receptor in the pituitary gland to suppress ovarian and testicular functions.

Specifications

Chemistry
Sequence one letter code
  • Ac-{d-A[3-(2-naphthyl)]}-[d-F(4-Cl)]-{d-A[3-(3-pyridyl)]}-SY-(d-Cit)-LRP-d-A-NH2•Acetate
Sequence three letter code
  • Ac-{D-Ala[3-(2-naphthyl)]}-[D-Phe(4-Cl)]-{D-Ala[3-(3-pyridyl)]}-Ser-Tyr-(D-Cit)-Leu-Arg-Pro-D-Ala-NH2 • Acetate
CAS registry number
  • 120287-85-6
Molecular Formula
  • C70H92ClN17O14
Molecular Mass/ Weight
  • 1431.2•60
Modification
Conjugation
  • Unconjugated
Quantity & Purity
Purity
  • Peak Area by HPLC ≥95%
Storage & stability
Form
  • Lyophilized
Storage Conditions
  • - 20 °C
Activity
Biomarker Target
Research Area
Sub-category Research Area
Usage
  • Research use
Source
Source / Species
  • Synthetic construct

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References

Luteinizing hormone-releasing hormone antagonist Cetrorelix regulates the expression of Gαs and Gαi protein subunits and adenylate cyclase activity in rat ovary, breast and pituitary

Intl J Oncol . 2004 Mar 01 ; 24(3) 725 | DOI : https://doi.org/10.3892/ijo.24.3.725

  • B. Collado
  • et al

Disposition and Metabolism of Cetrorelix, A Potent Luteinizing Hormone-Releasing Hormone Antagonist, in Rats and Dogs

Drug Metabolism and Disposition . 2000 Jan 01 ; 28(1) 10-20 | DOI : PMID: 10611134

  • M. Schwahn
  • et al