IMG-EN-AS-65487-01.jpg
Peptides

Protease-Activated Receptor-1, PAR-1 Antagonist 2, amide - 1 mg

$235.00
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  • Cat.Number : AS-65487
  • Availability :
    In production

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This peptide is a PAR-1 antagonist which inhibited SFLLRNP induced platelet aggregation with an IC50 of 115 uM. Antagonists specific for the thrombin receptor can be promising compounds for treatment of thrombosis.

Specifications

Chemistry
Sequence one letter code
  • S-F(para-Fluoro)-Aad-LRNP-NH2
Sequence three letter code
  • Ser-parafluoroPhe-Aad-Leu-Arg-Asn-Pro-NH2
Molecular Mass/ Weight
  • 893
Modification
Conjugation
  • Unconjugated
Quantity & Purity
Purity
  • Peak Area by HPLC ≥95%
Storage & stability
Form
  • Lyophilized
Storage Conditions
  • - 20 °C
Activity
Biomarker Target
Research Area
Sub-category Research Area
Usage
  • Research use
Source
Source / Species
  • human

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References

Design and Synthesis of para-Fluorophenylalanine Amide Derivatives as Thrombin Receptor Antagonists

J Biochem . 1999 Jul 01 ; 126(1) 174 | DOI : https://doi.org/10.1093/oxfordjournals.jbchem.a022419

  • T. Fujita
  • et al